Bambuterol, a bronchodilator prodrug with sustained action, enhances delivery of active drug to the lung.
As exemplified with bambuterol, a bronchodilator prodrug with sustained action, increased therapeutic selectivity can be obtained as a result of altered tissue distribution and pharmacokinetics rather than of increased beta 2-adrenoceptor selectivity.
Mesh Terms:
Animals, Asthma, Bronchodilator Agents, Guinea Pigs, Humans, In Vitro Techniques, Lung, Prodrugs, Terbutaline, Tissue Distribution
Animals, Asthma, Bronchodilator Agents, Guinea Pigs, Humans, In Vitro Techniques, Lung, Prodrugs, Terbutaline, Tissue Distribution
Agents Actions Suppl.
Date: Jan. 01, 1988
PubMed ID: 3262993
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