small molecule

Azatadine

Synonyms/Brands: Azatadin, Azatadina, Azatadine, Azatadinum, optimine tab, trinalin repetabs, 6,11-Dihydro-11-(1-methyl-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-b)pyridine, 11-(1-Methyl-4-piperidinylidene)-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridine

Antihistamines such as azatadine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihistamines antagonize those pharmacological effects of histamine which are mediated through activation of H1- receptor sites and thereby reduce the intensity of allergic reactions and tissue injury response involving histamine release.

Molecular Formula: C₂₀H₂₂N₂

Molecular Weight:: 290.4021

CAS:: 3964-81-6

ATC:: R06AX09

InChiKey:: SEBMTIQKRHYNIT-UHFFFAOYSA-N

InChi:: InChI=1S/C20H22N2/c1-22-13-10-16(11-14-22)19-18-7-3-2-5-15(18)8-9-17-6-4-12-21-20(17)19/h2-7,12H,8-11,13-14H2,1H3

SMILES:: CN1CCC(CC1)=C1C2=CC=CC=C2CCC2=C1N=CC=C2

IUPAC Name:: 2-(1-methylpiperidin-4-ylidene)-4-azatricyclo[9.4.0.0,]pentadeca-1(15),3(8),4,6,11,13-hexaene

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709

Interactors 1
Chemical Interactions 5
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Chemical Summary

Azatadine