BAIT

SMO

FZD11, Gx, SMOH
smoothened, frizzled class receptor
Homo sapiens

Co-crystal Structure

Interaction directly demonstrated at the atomic level by X-ray crystallography. Also used for NMR or Electron Microscopy (EM) structures. If there is no obvious bait-hit directionality to the interaction involving 3 or more proteins, then the co-crystallized proteins should be listed as a complex.

Publication

Cryo-EM structure of oxysterol-bound human Smoothened coupled to a heterotrimeric Gi.

Qi X, Liu H, Thompson B, McDonald J, Zhang C, Li X

The oncoprotein Smoothened (SMO), a G-protein-coupled receptor (GPCR) of the Frizzled-class (class-F), transduces the Hedgehog signal from the tumour suppressor Patched-1 (PTCH1) to the glioma-associated-oncogene (GLI) transcription factors, which activates the Hedgehog signalling pathway1,2. It has remained unknown how PTCH1 modulates SMO, how SMO is stimulated to form a complex with heterotrimeric G proteins and whether G-protein coupling contributes to ... [more]

Nature Dec. 01, 2018; 571(7764);279-283 [Pubmed: 31168089]

Throughput

  • Low Throughput

Curated By

  • BioGRID